Lessons learned from the development of kinase inhibitors Journal Article


Author: Sawyers, C. L.
Article Title: Lessons learned from the development of kinase inhibitors
Keywords: vasculotropin; cancer survival; unclassified drug; gene mutation; clinical trial; drug tolerability; sorafenib; erlotinib; sunitinib; patient selection; drug targeting; animals; imatinib; melanoma; enzyme inhibition; breast cancer; gene expression profiling; protein kinase inhibitor; epidermal growth factor receptor 2; lung cancer; high throughput screening; drug screening; drug resistance, neoplasm; drug discovery; enzyme activity; abelson kinase; dasatinib; chronic myeloid leukemia; drug selectivity; mutational analysis; protein kinase inhibitors; patient care; drug research; dna; mammalian target of rapamycin; malignant neoplastic disease; dna sequence; antiinflammatory activity; pharmacogenetics; bcr abl protein; robotics; trastuzumab; nilotinib; protein kinase; b raf kinase; rapamycin; drug protein binding; scatter factor receptor; drug indication; plx 4032; drug industry; individualization; kidney graft rejection; kidney transplantation
Journal Title: Clinical Advances in Hematology & Oncology
Volume: 7
Issue: 9
ISSN: 1543-0790
Publisher: Millennium Medical Publishing, Inc  
Date Published: 2009-09-01
Start Page: 588
End Page: 589
Language: English
PUBMED: 20020670
PROVIDER: scopus
DOI/URL:
Notes: --- - "Export Date: 30 November 2010" - "Source: Scopus"
Citation Impact
MSK Authors
  1. Charles L Sawyers
    225 Sawyers