53 Results

People

  1. Danishefsky
    Danishefsky
  2. Chou
    Chou
  3. Stachel
    Stachel
  4. Chappell
    Chappell
  5. Fornier
    Fornier
  6. Lee
    Lee
  7. Balog
    Balog
  8. Rivkin
    Rivkin
  9. Spriggs
    Spriggs
  10. Zhang
    Zhang

Groups

  1. Molecular Pharmacology and Chemistry Program Faculty (29)
  2. Sloan Kettering Institute Faculty (29)
  3. Department of Medicine (20)
  4. Solid Tumor Oncology Division (19)
  5. Breast Medicine Service (10)
  6. Survivorship Research (8)
  7. Sloan Kettering Institute Postdocs (7)
  8. Genitourinary Oncology Service (6)
  9. Biostatistics Service (4)
  10. Epidemiology and Biostatistics (4)
  1. "epothilones"
Formats
  1. Journal Article (52)
  2. Book Section (1)
Groups
  1. Molecular Pharmacology and Chemistry Program Faculty (29)
  2. Sloan Kettering Institute Faculty (29)
  3. Department of Medicine (20)
  4. Solid Tumor Oncology Division (19)
  5. Breast Medicine Service (10)
  6. Survivorship Research (8)

More Groups

People
  1. Samuel Danishefsky (29)
  2. Ting-Chao Chou (20)
  3. Shawn Stachel (8)
  4. Chul Lee (7)
  5. Mark Chappell (7)
  6. Monica Fornier (7)

More People

Years
  1. 2013 (1)
  2. 2012 (3)
  3. 2010 (3)
  4. 2009 (4)
  5. 2008 (3)
  6. 2007 (8)

More Years

Publications
  1. Proceedings of the National Academy of Sciences of the United States of America (7)
  2. Angewandte Chemie - International Edition (5)
  3. Journal of Clinical Oncology (5)
  4. Investigational New Drugs (4)
  5. Journal of Organic Chemistry (4)
  6. Journal of the American Chemical Society (4)

More Publications

Publishers
  1. American Chemical Society (10)
  2. Wiley Blackwell (9)
  3. National Academy of Sciences (7)
  4. American Society of Clinical Oncology (5)
  5. American Association for Cancer Research (4)
  6. Springer (4)

More Publishers

Results (53)


Citation style sort is year ascending, and then by author or title. Author ascending is default.
  • Synthesis and conformational analysis of (E)-9,10-dehydroepothilone B: A suggestive link between the chemistry and biology of epothilones
    Journal Article

    Yoshimura, F.; Rivkin, A.; Gabarda, A. E.; Chou, T. C.; Dong, H.; Sukenick, G.; Morel, F. F.; Taylor, R. E.; Danishefsky, S. J.
    Angewandte Chemie - International Edition (2003)

    Fulltext@MSK | Save
  • Pilot study of epothilone B analog (BMS-247550) and estramustine phosphate in patients with progressive metastatic prostate cancer following castration
    Journal Article

    Smaletz, O.; Galsky, M.; Scher, H. I.; Delacruz, A.; Slovin, S. F.; Morris, M. J.; Solit, D. B.; Davar, U.; Schwartz, L.; Kelly, W. K.
    Annals of Oncology (2003)

    Fulltext@MSK | Save
  • Complex target-oriented total synthesis in the drug discovery process: The discovery of a highly promising family of second generation epothilones
    Journal Article

    Rivkin, A.; Yoshimura, F.; Gabarda, A. E.; Chou, T. C.; Dong, H.; Tong, W. P.; Danishefsky, S. J.
    Journal of the American Chemical Society (2003)

    Fulltext@MSK | Save
  • Design and total synthesis of a superior family of epothilone analogues, which eliminate xenograft tumors to a nonrelapsable state
    Journal Article

    Chou, T. C.; Dong, H.; Rivkin, A.; Yoshimura, F.; Gabarda, A. E.; Cho, Y. S.; Tong, W. P.; Danishefsky, S. J.
    Angewandte Chemie - International Edition (2003)

    Fulltext@MSK | Save
  • Total syntheses of [17]- and [18]dehydrodesoxyepothilones B via a concise ring-closing metathesis-based strategy: Correlation of ring size with biological activity in the epothilone series
    Journal Article

    Rivkin, A.; Njardarson, J. T.; Biswas, K.; Chou, T. C.; Danishefsky, S. J.
    Journal of Organic Chemistry (2002)

    Fulltext@MSK | Save
  • Probing the SAR of dEpoB via chemical synthesis: A total synthesis evaluation of C26-(1,3-dioxolanyl)-12,13-desoxyepothilone B
    Journal Article

    Chappell, M. D.; Harris, C. R.; Kuduk, S. D.; Balog, A.; Wu, Z.; Zhang, F.; Lee, C. B.; Stachel, S. J.; Danishefsky, S. J.; Chou, T. C.; more...
    Journal of Organic Chemistry (2002)

    Fulltext@MSK | Save
  • Highly concise routes to epothilones: The total synthesis and evaluation of epothilone 490
    Journal Article

    Biswas, K.; Lin, H.; Njardarson, J. T.; Chappell, M. D.; Chou, T. C.; Guan, Y.; Tong, W. P.; He, L.; Horwitz, S. B.; Danishefsky, S. J.
    Journal of the American Chemical Society (2002)

    Fulltext@MSK | Save
  • Chemical synthesis and biological studies of the epothilones - Microtubule stabilizing agents with enhanced activity against multidrug-resistant cell lines and tumors
    Book Section

    Harris, C. R.; Kuduk, S. D.; Danishefsky, S. J.
    In Keinan, E.; Schechter, I. (Eds.) Chemistry for the 21st Century (2001)

    Fulltext@MSK | Save
  • The synthesis, discovery, and development of a highly promising class of microtubule stabilization agents: Curative effects of desoxyepothilones B and F against human tumor xenografts in nude mice
    Journal Article

    Chou, T. C.; O'Connor, O. A.; Tong, W. P.; Guan, Y.; Zhang, Z. G.; Stachel, S. J.; Lee, C.; Danishefsky, S. J.
    Proceedings of the National Academy of Sciences of the United States of America (2001)

    Fulltext@MSK | Save
  • Insights into long-range structural effects on the stereochemistry of aldol condensations: A practical total synthesis of desoxyepothilone F
    Journal Article

    Lee, C. B.; Wu, Z.; Zhang, F.; Chappell, M. D.; Stachel, S. J.; Chou, T. C.; Guan, Y.; Danishefsky, S. J.
    Journal of the American Chemical Society (2001)

    Fulltext@MSK | Save